Bilcer, Geoffrey: search on Z-Library

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1

Structure-based design of cycloamide–urethane-derived novel inhibitors of human brain memapsin 2 (β-secretase)

Arun K. Ghosh, Thippeswamy Devasamudram, Lin Hong, Christopher DeZutter, Xiaoming Xu, Vajira Weerasena, Gerald Koelsch, Geoffrey Bilcer, Jordan Tang

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2005

Language:

english

File:

PDF, 374 KB

english, 2005

2

In vivo inhibition of Aβ production by memapsin 2 (β-secretase) inhibitors

Wan-Pin Chang, Gerald Koelsch, Stephen Wong, Deborah Downs, Huining Da, Vajira Weerasena, Brian Gordon, Thippeswamy Devasamudram, Geoffrey Bilcer, Arun K. Ghosh, Jordan Tang

Journal:

Journal of Neurochemistry

Year:

2004

Language:

english

File:

PDF, 336 KB

english, 2004

3

A stereoselective synthesis of (+)-boronolide

Arun K Ghosh, Geoffrey Bilcer

Journal:

Tetrahedron Letters

Year:

2000

Language:

english

File:

PDF, 107 KB

english, 2000

4

Structure-Based Design: Potent Inhibitors of Human Brain Memapsin 2 (β-Secretase)

Ghosh, Arun K., Bilcer, Geoffrey, Harwood, Cynthia, Kawahama, Reiko, Shin, Dongwoo, Hussain, Khaja Azhar, Hong, Lin, Loy, Jeffrey A., Nguyen, Chan, Koelsch, Gerald, Ermolieff, Jacques, Tang, Jordan

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 121 KB

english, 2001

5

P4-374 In vivo inhibition of brain Aβ level by memapsin 2 (β-secretase) inhibitors

Chang, Wan-Pin, Koelsch, Gerald, Wong, Stephen, Downs, Deborah, Da, Huining, Weerasena, Vajira, Gordon, Brian, Devasamudram, Thippeswamy, Bilcer, Geoffrey, Ghosh, Arun K., Tang, Jordan

Journal:

Neurobiology of Aging

Year:

2004

Language:

english

File:

PDF, 166 KB

english, 2004

6

The Microtubule Stabilizing Agent Laulimalide Does Not Bind in the Taxoid Site, Kills Cells Resistant to Paclitaxel and Epothilones, and May Not Require Its Epoxide Moiety for Activity †

Pryor, Donald E., O'Brate, Aurora, Bilcer, Geoffrey, Díaz, J. Fernando, Wang, Yuefang, Wang, Yong, Kabaki, Mikio, Jung, M. Katherine, Andreu, José M., Ghosh, Arun K., Giannakakou, Paraskevi, Hamel, Er

Journal:

Year:

2002

Language:

english

File:

PDF, 138 KB

english, 2002

7

Structure-based design, synthesis and biological evaluation of novel β-secretase inhibitors containing a pyrazole or thiazole moiety as the P3 ligand

Ghosh, Arun K., Brindisi, Margherita, Yen, Yu-Chen, Xu, Xiaoming, Huang, Xiangping, Devasamudram, Thippeswamy, Bilcer, Geoffrey, Lei, Hui, Koelsch, Gerald, Mesecar, Andrew D., Tang, Jordan

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2015

Language:

english

File:

PDF, 1.58 MB

english, 2015

8

Real-time Microdialysis for aβ Inhibition And Pk/pd Analysis in A Nonhuman Primate Model: In Vivo Efficacy of a Bace-1 Inhibitor

Yu, Jeremy, Koelsch, Gerald, Li, Aiqun, Turner, Robert T., Bilcer, Geoffrey M., Miyake, Akira, Hamakawa, Nozomu, Terashita, Shigeyuki, Matsuoka, Nobuya, Hey, John A.

Journal:

Alzheimer's & Dementia

Year:

2010

Language:

english

File:

PDF, 45 KB

english, 2010

9

Design, Synthesis and X-ray Structure of Protein−Ligand Complexes: Important Insight into Selectivity of Memapsin 2 (β-Secretase) Inhibitors

Ghosh, Arun K., Kumaragurubaran, Nagaswamy, Hong, Lin, Lei, Hui, Hussain, Khaja Azhar, Liu, Chun-Feng, Devasamudram, Thippeswamy, Weerasena, Vajira, Turner, Robert, Koelsch, Gerald, Bilcer, Geoffrey,

Journal:

Journal of the American Chemical Society

Year:

2006

Language:

english

File:

PDF, 81 KB

english, 2006

10

ChemInform Abstract: A Stereoselective Synthesis of (+)-Boronolide.

Arun K. Ghosh, Geoffrey Bilcer

Journal:

Year:

2000

File:

PDF, 33 KB

2000

11

APN1125: A NOVEL A7 NICOTINIC ACETYLCHOLINE RECEPTOR PARTIAL AGONIST

Koelsch, Gerald, Meltzer, Leonard T., Yoshimura, Ryan F., Terry, Alvin V., Callahan, Patrick M., Bilcer, Geoffrey, Ng, John, Ng, Raymond, Gee, Kelvin W., Kelly, Terence A.

Journal:

Alzheimer's & Dementia

Year:

2014

Language:

english

File:

PDF, 58 KB

english, 2014

12

Memapsin 2 (Beta-Secretase) Inhibitor Drug, between Fantasy and Reality

Ghosh, Arun, Bilcer, Geoffrey, Hong, Lin, Koelsch, Gerald, Tang, Jordan

Journal:

Current Alzheimer Research

Year:

2007

Language:

english

File:

PDF, 186 KB

english, 2007

13

ChemInform Abstract: Syntheses of FDA Approved HIV Protease Inhibitors

Arun K. Ghosh, Geoffrey Bilcer, Gary Schiltz

Journal:

Year:

2002

File:

PDF, 24 KB

2002

14

Tartaric Acid and Tartrates in the Synthesis of Bioactive Molecules

Ghosh, Arun K., Koltun, Elena S., Bilcer, Geoffrey

Journal:

Year:

2001

Language:

english

File:

PDF, 1.85 MB

english, 2001

15

In vivo efficacy of BACE-1 inhibitor CTS21166 (ASP1702) in rat CNS compartments

Yu, Jeremy, Koelsch, Gerald, Li, Aiqun, Turner, Robert T., Bilcer, Geoffrey M., Grove, Carl, Hsu, Henry H., Shitaka, Yoshitsugu, Hamakawa, Nozomu, Terashita, Shigeyuki, Matsuoka, Nobuya, Tang, Jordan,

Journal:

Alzheimer's & Dementia

Year:

2009

Language:

english

File:

PDF, 62 KB

english, 2009

16

APN0417: A potent and efficacious α7 nAChR positive allosteric modulator

Dasse, Olivier, Bilcer, Geoffrey, Putman, David, Ng, Raymond, Gee, Kelvin, Stevens, Karen E., Tran, Minhtam, Johnstone, Tim, Yoshimura, Ryan F., Koelsch, Gerald, Kelly, Terence A.

Journal:

Biochemical Pharmacology

Year:

2015

Language:

english

File:

PDF, 149 KB

english, 2015

17

Syntheses of FDA Approved HIV Protease Inhibitors

Ghosh, Arun K., Bilcer, Geoffrey, Schiltz, Gary

Journal:

Year:

2001

Language:

english

File:

PDF, 1.11 MB

english, 2001

18

Design, Synthesis, and X-ray Structure of Potent Memapsin 2 (β-Secretase) Inhibitors with Isophthalamide Derivatives as the P 2- P 3 -Ligands

Ghosh, Arun K., Kumaragurubaran, Nagaswamy, Hong, Lin, Kulkarni, Sarang S., Xu, Xiaoming, Chang, Wanpin, Weerasena, Vajira, Turner, Robert, Koelsch, Gerald, Bilcer, Geoffrey, Tang, Jordan

Journal:

Journal of Medicinal Chemistry

Year:

2007

Language:

english

File:

PDF, 269 KB

english, 2007

19

ChemInform Abstract: Tartaric Acid and Tartrates in the Synthesis of Bioactive Molecules

Arun K. Ghosh, Elena S. Koltun, Geoffrey Bilcer

Journal:

Year:

2001

File:

PDF, 24 KB

2001

20

APN1125: A clinical stage α7 nicotinic acetylcholine receptor partial agonist

Koelsch, Gerald, Detke, Michael J., Stevens, Karen E., Meltzer, Leonard T., Terry, Alvin V., Callahan, Patrick M., Yoshimura, Ryan F., Bilcer, Geoffrey, Anderson, Paul C., Ng, John, Ng, Raymond, Kelly

Journal:

Biochemical Pharmacology

Year:

2015

Language:

english

File:

PDF, 150 KB

english, 2015

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